From: Targeting multidrug resistance in cancer by natural chemosensitizers
Targeted ABC transporter | Chemosensitizer | Reference |
---|---|---|
ABCB1/P-gp/MDR-1 | 5-Bromotetrandrine | (Jin et al. 2005) |
Abietane diterpene | (Madureira et al. 2004a) | |
Alisol B 23-acetate | (Wang et al. 2004a) | |
Amooranin | (Ramachandran et al. 2003) | |
Baicalein and derivatives | (Lee et al. 2004) | |
Biochanin A | (Zhang and Morris 2003) | |
Bitter melon extract | (Limtrakul et al. 2004) | |
Bufalin | (Mahringer et al. 2010) | |
Cannabinoids | ||
β-Carotene | (Teng et al. 2016) | |
Catechins | (Kitagawa et al. 2004) | |
Cepharanthine | (Koizumi et al. 1995) | |
Coumarins | (Raad et al. 2006) | |
Curcumin and semisynthetic derivatives | (Chearwae et al. 2004; Anuchapreeda et al. 2002; Ooko et al. 2016) | |
Cycloartanes | (Madureira et al. 2004b) | |
Deoxyschizandrin | (Yoo et al. 2007) | |
Didehydrostemofolines | (Umsumarng et al. 2017) | |
Eudesmin | (Lim et al. 2007) | |
Euphocharacins A-L | (Corea et al. 2004) | |
Ginkgo biloba extract | ||
Ginsenoside Rg | (Kim et al. 2003) | |
Grapefruit juice extracts | (de Castro et al. 2007) | |
Hapalosin | (Palomo et al. 2004) | |
Hypericin and hyperforin | (Wang et al. 2004b) | |
Isoquinoline alkaloid, isotetrandrine | (Wang and Yang 2008) | |
Isostemofoline | (Umsumarng et al. 2017) | |
Jatrophanes | ||
Kaempferia parviflora extracts | (Patanasethanont et al. 2007a) | |
Kavalactones | (Weiss et al. 2005) | |
Morin | (Zhang and Morris 2003) | |
Ningalin B and derivatives | ||
Opiates | (Hemauer et al. 2009) | |
Phloretin | (Zhang and Morris 2003) | |
Piperine | (Han et al. 2008) | |
Polyoxypregnanes | (KKW et al. 2017) | |
Protopanaxatriol ginsenosides | (Choi et al. 2003) | |
Pyranocoumarins | (Wu et al. 2003) | |
Quercetin | ||
Schisandrol A | (Fong et al. 2007) | |
Sesquiterpenes | (Munoz-Martinez et al. 2004) | |
Silymarin | (Zhang and Morris 2003) | |
Sinensetin | (Choi et al. 2002) | |
Stemona curtisii root extract | (Limtrakul et al. 2007a) | |
Taxane derivatives | ||
Terpenoids | (Yoshida et al. 2006) | |
Tetrandine | (Fu et al. 2004) | |
Vitamin E TPGS | (Collnot et al. 2007) | |
ABCG2/BCRP/MXR | 3′-4′-7-Trimethoxyflavone | (Katayama et al. 2007) |
6-Prenylchrysin | (Ahmed-Belkacem et al. 2005) | |
Acacetin | (Imai et al. 2004) | |
Biochanin A | (Zhang et al. 2004) | |
Cannabinoids | (Holland et al. 2007) | |
Chrysin | (Zhang et al. 2004) | |
Curcumin | (Chearwae et al. 2006a) | |
Daizein | (Cooray et al. 2004) | |
Eupatin | (Henrich et al. 2006) | |
Genistein | (Imai et al. 2004) | |
Ginsenosides | (Jin et al. 2006) | |
Harmine | (Ma and Wink 2010) | |
Hesperetin | (Cooray et al. 2004) | |
Kaempferol | (Imai et al. 2004) | |
Naringenin | (Imai et al. 2004) | |
Plumbagin | (Shukla et al. 2007) | |
Quercetin | (Cooray et al. 2004) | |
Resveratrol | (Cooray et al. 2004) | |
Rotenoids | (Ahmed-Belkacem et al. 2007) | |
Silymarin | (Cooray et al. 2004) | |
Stilbenoids | (Morita et al. 2005) | |
Tectochrysin | (Ahmed-Belkacem et al. 2005) | |
Terpenoids | (Yoshida et al. 2008) | |
Tetrahydrocurcumin | (Limtrakul et al. 2007b) | |
ABCC1/MRP1 | Cannabinoids | (Holland et al. 2008) |
Cepharanthine | (Abe et al. 1995) | |
Curcumin | (Chearwae et al. 2006b) | |
Ginkgo biloba extract | (Nabekura et al. 2008) | |
Kaempferia parviflora extracts | (Patanasethanont et al. 2007b) | |
Myricetin | (van Zanden et al. 2005) | |
Quercetin | ||
Stemona curtisii root extract | (Limtrakul et al. 2007a) |